发明名称 |
Peripherally selective piperidine carboxylate opioid antagonists |
摘要 |
3,4,4-trisubstitutedpiperidinyl-N-alkylcarboxylates and intermediates for their preparation are provided. These piperidine-N-alkylcarboxylates are useful as peripheral opioid antagonists.
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申请公布号 |
US5250542(A) |
申请公布日期 |
1993.10.05 |
申请号 |
US19920916783 |
申请日期 |
1992.07.17 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
CANTRELL, BUDDY E.;ZIMMERMAN, DENNIS M. |
分类号 |
C07D211/34;C07D405/12;C07D413/12;(IPC1-7):A61K31/445;C07D401/12;C07D211/32 |
主分类号 |
C07D211/34 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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