发明名称 |
Direct esterification of mycophenolic acid |
摘要 |
Mycophenolate mofetil is made non-catalytically by refluxing mycophenolic acid with 2-morpholinoethanol in an inert organic solvent capable of azeotropic removal of water.
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申请公布号 |
US5247083(A) |
申请公布日期 |
1993.09.21 |
申请号 |
US19920993146 |
申请日期 |
1992.12.18 |
申请人 |
SYNTEX (U.S.A.) INC. |
发明人 |
KNOX, MARTIN;DONEGAN, GREGORY;SMITH, DENNIS A. |
分类号 |
C07D307/88 |
主分类号 |
C07D307/88 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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