发明名称 PROCEDIMIENTO DE PREPARACION DE DERIVADOS DE [(BENZOIMIDAZOL-1-IL)-QUINOLIN-8-IL]-PIPERIDIN-4-ILAMINA, UTILES EN EL TRATAMIENTO DEL CRECIMIENTO CELULAR ANORMAL, POR DESPROTECCION DEL GRUPO BOC CON UN ALCOXIDO DE METAL EN PRESENCIA DE UN EQUIVALENTE D
摘要 The present invention relates to a process for preparing a compound of the formula I or a pharmaceutically acceptable salt, prodrug, hydrate or solvate thereof, wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3 </SUP>and R<SUP>4 </SUP>are as defined herein. The compound of formula I is useful in the treatment of abnormal cell growth, such as cancer, in mammals.
申请公布号 CL2004001470(A1) 申请公布日期 2005.05.13
申请号 CL20040001470 申请日期 2004.06.14
申请人 PFIZER PRODUCTS INC. 发明人 NORMA JACQUELINE TOM, DAVID HAROLD BROWN RIPIN,MICHAEL JAMES CASTALDI
分类号 A61K31/47;A61K31/4709;C07D211/00;C07D215/12;C07D215/38;C07D235/02;C07D305/06;C07D401/14;C07D405/14;(IPC1-7):A61K31/47 主分类号 A61K31/47
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