发明名称 N-ARYL-N1-AZABICYCLO-UREAS AS 5-HT3 ANTAGONISTS
摘要 Compounds of formula (I) and pharmaceutically acceptable salts thereof, wherein A1, A2, A3 and the carbon atoms to which they are attached form a 5- or 6-membered non-aromatic heterocyclic ring containing at least one -O-, -CO- or -N-; R1 and R2 are hydrogen or C1-6 alkyl; Y is hydrogen, halo, C1-6 alkyl or C1-6 alkoxy; L is O or NH; Z is an azabicyclic side chain; having 5-HT3 receptor antagonist activity.
申请公布号 WO9308185(A1) 申请公布日期 1993.04.29
申请号 WO1992GB01876 申请日期 1992.10.13
申请人 SMITHKLINE BEECHAM PLC 发明人 KING, FRANCIS, DAVID;GASTER, LARAMIE, MARY
分类号 C07D451/04;C07D498/08 主分类号 C07D451/04
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