| 摘要 |
PCT No. PCT/US91/08850 Sec. 371 Date Jul. 26, 1993 Sec. 102(e) Date Jul. 26, 1993 PCT Filed Nov. 25, 1991 PCT Pub. No. WO92/09297 PCT Pub. Date Jun. 11, 1992.Peptide mimics, having a constrained peptide backbone conformation, are HIV protease inhibitors. A compound of this invention is, for example, 3-Benzyl-5(alaninyl-1-aminoethyl)-2,3,6,7-tetrahydro-N-azepinyl-2-propionyl-valinyl-valinyl methyl ester. |
