发明名称 |
Phosphorylating agent and method for forming phosphodiester bond using the same. |
摘要 |
<p>A phosphorylating agent represented by the following general formula [1]: <CHEM> wherein R represents a protective group of the phosphoric acid; and X represents a heterocyclic residue represented by the following general formula [2]: <CHEM> wherein Y represents a single bond or an oxygen or sulfur atom; Z represents a heterocyclic nucleus comprising at least one nitrogen atom as a ring-forming element and may be condensed with another aromatic ring; and W represents one or more substituents other than a hydrogen atom. The phosphorylating agent is stable, can rapidly proceed phosphodiester bond-forming reactions in good selectivity under mild conditions and thus makes it possible to perform a reaction even in a relatively large scale.</p> |
申请公布号 |
EP0483732(A2) |
申请公布日期 |
1992.05.06 |
申请号 |
EP19910118365 |
申请日期 |
1991.10.28 |
申请人 |
FUJI PHOTO FILM CO., LTD. |
发明人 |
MORI, HIDETO |
分类号 |
C07B47/00;C07F9/09;C07F9/12;C07F9/6515;C07F9/6518;C07F9/6524;C07F9/6527;C07F9/653;C07F9/655 |
主分类号 |
C07B47/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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