发明名称 |
PROCESS FOR PRODUCING DIACYL DERIVATIVES OF RIFAMYCINS SUBSTITUTED WITH 4-(TRIALKYLBENZYL)-PIPERAZINYL GROUP AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME |
摘要 |
Acylated 3-piperazinyl-substd. rifamycin derivs. of formula (I) and their salts are new: R= lower alkyl; R1= tri(lower alkyl) methylcarbonyl; one of R2 and R3 = tri (lower alkyl) methylcarbonyl and the other is H. - More specifically R=Me; R1 and one of R2and R3 = pivaloyl; the other is H. |
申请公布号 |
HU201555(B) |
申请公布日期 |
1990.11.28 |
申请号 |
HU19870004776 |
申请日期 |
1987.09.25 |
申请人 |
CIBA GEIGY AG |
发明人 |
TRAXLER PETER;MUELLER KLAUS;KUMP WILHELM |
分类号 |
A61K31/495;C07D498/08 |
主分类号 |
A61K31/495 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|