发明名称 FLUOROCYTIDINE DERIVATIVES, THEIR PREPARATION AND MEDICAL PREPARATIONS CONTAINING THEM
摘要 <p>derivs. of formula (I), their hydrates and solvates are new. In (I) R1, R2 and R3 = H or a gp. which is easily removed under physiological conditions, at least one of them being other than H. Specifically easily hydrolysed gps. are of formulae R4CO, R5O.CO or R6S.CO; R4 = H, alkyl, cycloalkyl, oxoalkyl, alkenyl, aralkyl or aryl; R5 and R6 = alkyl or aralkyl.</p>
申请公布号 EP0316704(A3) 申请公布日期 1990.11.22
申请号 EP19880118515 申请日期 1988.11.07
申请人 F. HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT 发明人 FUJIU, MORIO;ISHITSUKA, HIDEO;MIWA, MASANORI;UMEDA, ISAO IMPERIAL HIGASHIHAKURAKU;YOKOSE, KAZUTERU
分类号 C07H19/06;(IPC1-7):C07H19/067;A61K31/70 主分类号 C07H19/06
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