发明名称 |
FLUOROCYTIDINE DERIVATIVES, THEIR PREPARATION AND MEDICAL PREPARATIONS CONTAINING THEM |
摘要 |
<p>derivs. of formula (I), their hydrates and solvates are new. In (I) R1, R2 and R3 = H or a gp. which is easily removed under physiological conditions, at least one of them being other than H. Specifically easily hydrolysed gps. are of formulae R4CO, R5O.CO or R6S.CO; R4 = H, alkyl, cycloalkyl, oxoalkyl, alkenyl, aralkyl or aryl; R5 and R6 = alkyl or aralkyl.</p> |
申请公布号 |
EP0316704(A3) |
申请公布日期 |
1990.11.22 |
申请号 |
EP19880118515 |
申请日期 |
1988.11.07 |
申请人 |
F. HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT |
发明人 |
FUJIU, MORIO;ISHITSUKA, HIDEO;MIWA, MASANORI;UMEDA, ISAO IMPERIAL HIGASHIHAKURAKU;YOKOSE, KAZUTERU |
分类号 |
C07H19/06;(IPC1-7):C07H19/067;A61K31/70 |
主分类号 |
C07H19/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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