发明名称 |
Process for the synthesis of alpha n alkylated amino acids and esters thereof, application to the synthesis of carboxyalkyl dipeptides |
摘要 |
Stereoselective process for the industrial synthesis of compounds of formula (I): <IMAGE> (I) where R1 is linear or branched lower alkyl with 1 to 6 carbon atoms, R2 is a linear or branched lower alkyl with 1 to 4 carbon atoms, employing inexpensive starting materials and obtaining optimum yields. Application to the synthesis of carboxyalkyl dipeptides.
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申请公布号 |
US4902817(A) |
申请公布日期 |
1990.02.20 |
申请号 |
US19880245353 |
申请日期 |
1988.09.16 |
申请人 |
ADIR ET CIE |
发明人 |
VINCENT, MICHEL;BALIARDA, JEAN;MARCHAND, BERNARD;REMOND, GEORGES |
分类号 |
C07D209/12;A61K31/395;A61K31/40;A61K31/403;A61K31/4035;A61K31/404;A61K31/435;A61K31/47;A61K31/472;A61P3/00;A61P9/00;A61P9/12;B01J23/40;B01J23/755;C07B31/00;C07B53/00;C07B61/00;C07C67/00;C07C227/00;C07C227/18;C07C227/32;C07C227/42;C07C229/16;C07D209/14;C07D209/42;C07D209/44;C07D209/52;C07D215/14;C07D217/16;C07D221/22;C07D453/06;C07K5/02 |
主分类号 |
C07D209/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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