发明名称 Process for the synthesis of alpha n alkylated amino acids and esters thereof, application to the synthesis of carboxyalkyl dipeptides
摘要 Stereoselective process for the industrial synthesis of compounds of formula (I): <IMAGE> (I) where R1 is linear or branched lower alkyl with 1 to 6 carbon atoms, R2 is a linear or branched lower alkyl with 1 to 4 carbon atoms, employing inexpensive starting materials and obtaining optimum yields. Application to the synthesis of carboxyalkyl dipeptides.
申请公布号 US4902817(A) 申请公布日期 1990.02.20
申请号 US19880245353 申请日期 1988.09.16
申请人 ADIR ET CIE 发明人 VINCENT, MICHEL;BALIARDA, JEAN;MARCHAND, BERNARD;REMOND, GEORGES
分类号 C07D209/12;A61K31/395;A61K31/40;A61K31/403;A61K31/4035;A61K31/404;A61K31/435;A61K31/47;A61K31/472;A61P3/00;A61P9/00;A61P9/12;B01J23/40;B01J23/755;C07B31/00;C07B53/00;C07B61/00;C07C67/00;C07C227/00;C07C227/18;C07C227/32;C07C227/42;C07C229/16;C07D209/14;C07D209/42;C07D209/44;C07D209/52;C07D215/14;C07D217/16;C07D221/22;C07D453/06;C07K5/02 主分类号 C07D209/12
代理机构 代理人
主权项
地址