发明名称 PROCESS FOR PRODUCTION OF CEFALOSPORIN-SALTS AND INJECTABLE COMPOSITIONS CONTAINING THEM AS ACTIVE SOBSTANCE
摘要 Temp. stable crystalline salts of alpha-(2-aminothiazol-4- yl) alpha-(Z)-methoxyiminoacetamido) -3 -(1-methyl-1-pyrrolidinio) methyl)-3-cephem-4-carboxylate (I) are claimed, selected from sulphuric, di-nitric, monohydrochloric and di-hydrochloric acid addn. salts and orthophosphoric acid addn. salts contg. 1.5-2 molar equivalents of H3PO4, or solvates of tehse. The salt may be mixed with a base e.g. L(+) lysine or L(+) arginine.
申请公布号 HUT50347(A) 申请公布日期 1990.01.29
申请号 HU19890000185 申请日期 1989.01.18
申请人 BRISTOL MYERS CO,US 发明人 KAPLAN,MURRAY A.,US;HUDYMA,ROBERT W.,US;LIPPER,ROBERT A.,US;SHIH, KUN M.,US;BOETTGER,SUSAN D.,US
分类号 C07D501/00;A61K31/40;A61K31/425;A61K31/545;A61K31/546;A61K47/00;A61K47/18;C07D;C07D501/04;C07D501/38;C07D501/46;C07D501/56;C07D501/60;(IPC1-7):C07D501/46 主分类号 C07D501/00
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