发明名称 6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives and intermediates therefor.
摘要 <p>This invention relates to novel 1,7-disubstituted-6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives and certain esters and cation salts thereof. This invention further relates to preparation of the compounds, antibacterial compositions containing the compounds and methods of using the compounds. This invention also relates to a novel process for preparing novel N-cyclopropyl intermediates useful for preparing certain of the 1,7-disubstituted-6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives of this invention which contain a cyclopropyl substituent at the 1 position as well as other 1,4-dihydroquinol-4-one-3-carboxylic acid derivatives so substituted with cyclopropyl.</p>
申请公布号 EP0348088(A1) 申请公布日期 1989.12.27
申请号 EP19890305969 申请日期 1989.06.13
申请人 PFIZER INC. 发明人 MCGUIRK, PAUL ROBERT
分类号 A61K31/47;A61P31/04;C07C211/52;C07C229/30;C07D215/56;C07D405/06 主分类号 A61K31/47
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