发明名称 ANALGESIC 1,2-BENZISOTHIAZOL-3-YLPIPERAZINE DERIVATIVES
摘要 <p>MJ-592 A series of non-oplate analgesics of Formula I wherein R1 is hydrogen, alkyl, aralkyl, or aryloxyalkyl; R2 is alkyl or hydrogen; and R3 and R4 are independently selected from hydrogen, alkyl, acyloxy, alkoxy, alkylthio, halogen, hydroxyl, or trifluoromethyl; or a pharmaceutically acceptable acid addition salt.</p>
申请公布号 CA1249587(A) 申请公布日期 1989.01.31
申请号 CA19850488887 申请日期 1985.08.16
申请人 BRISTOL-MYERS COMPANY 发明人 SMITH, DAVID W.;YEVICH, JOSEPH P.
分类号 A61K31/425;A61K31/428;A61K31/495;A61P25/02;A61P25/04;A61P25/20;C07D275/04;C07D319/00;C07D417/04;C07D417/12;(IPC1-7):C07D417/12;C07D417/14 主分类号 A61K31/425
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