发明名称 |
NYTT FOERFARANDE FOER FRAMSTAELLNING AV SOM LAEKEMEDEL ANVAENDBAR 4'-DEOXI-DAUNORUBICIN |
摘要 |
A new process for the preparation of the known 4'-deoxydaunorubicin and 4'-deoxydoxorubicin is disclosed. The used starting material is 4'-eip-N-trifluoroacetyldaunorubicin which is converted into 4'-deoxy-4'-iodo-N-trifluoroacetyl-daunorubicin from which 4'-deoxy-daunorubicin can be reductively obtained and eventually transformed, by known methods, into 4'-deoxy-doxorubicin. |
申请公布号 |
FI65997(B) |
申请公布日期 |
1984.04.30 |
申请号 |
FI19810002985 |
申请日期 |
1981.09.25 |
申请人 |
FARMITALIA CARLO ERBA S P A |
发明人 |
SUARATO ANTONIO;PENCO SERGIO;ARCAMONE FEDERICO |
分类号 |
C07D309/14;A61K31/65;C07H15/252;(IPC1-7):C07D309/14 |
主分类号 |
C07D309/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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