发明名称 GABA-ERGIC MODULATORS
摘要 FIELD: medicine. ^ SUBSTANCE: invention is related to new derivatives of benzoindazole of formula I , where radicals A1, A2, A3, R1, R2, R3, R4 and n have values mentioned in formula of invention, and their pharmaceutically acceptable salts, and also to application of these compounds for production of medicinal agent intended for modulation of 2-subsort of GABA receptor, and pharmaceutical composition that contains it. ^ EFFECT: application of compounds for preparation of medicinal agent intended for treatment of depression, disorder in the form of anxiety, psychic disorder, disturbed ability to learning and cognition, sleep disturbance, disorder in the form of cramps or fits or pain. ^ 16 cl, 5 tbl, 40 ex
申请公布号 RU2376292(C2) 申请公布日期 2009.12.20
申请号 RU20060107438 申请日期 2004.08.05
申请人 F.KHOFFMANN-LJA ROSH AG 发明人 LIN' SJAOFA;LOUKHED DEJVID GARRETT;NOVAKOVITS SANJA;O'JANG KAUND;PUTMAN DEJVID DZHORDZH;SOT MAJKL
分类号 A61K31/416;A61K31/4745;A61K31/519;A61P25/00;C07D231/56;C07D401/04;C07D401/12;C07D403/06;C07D405/04;C07D409/04;C07D413/12;C07D417/04;C07D471/02;C07D471/04;C07D487/02;C07D487/04 主分类号 A61K31/416
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