发明名称 3-(SUBSTITUTED) PROPENYLAMINOTHIAZOL-YLCEPHALOSPORANIC ACIDS AND ESTERS THEREOF
摘要 <p>This invention provides novel cephalosporanic acids and esters thereof having the general formula <IMAGE> wherein R2 is hydrogen, lower alkyl, lower alkenyl, lower alkynyl, cyclo(lower)alkyl or acyl, R3 is hydrogen, lower alkyl, lower alkoxy, lower alkanoyloxy, and R4 is hydrogen, pivaloyloxymethyl, acetoxymethyl, 1-acetoxyethyl, 5-methyl-2-oxo-1, 3-dioxolen-4-ylmethyl or 4-glycyloxybenzoyloxymethyl. These compounds, especially esters, are useful as broad spectrum antibiotics in the treatment and prevention of infectious diseases of mammals, and for other purposes known in the art.</p>
申请公布号 GR861611(B) 申请公布日期 1986.10.30
申请号 GR19860101611 申请日期 1986.06.20
申请人 BRISTOL-MYERS COMPANY 发明人 SEIJI LIMURA;YOSHIO ABE;OKUMURA JUN;TAKAYUKI NAITO;HAJIME KAMACHI
分类号 C07D501/20;A61K;A61K31/545;A61K31/546;A61P31/04;C07C;C07D;C07D277/28;C07D277/40;C07D277/42;C07D417/12;C07D501/00;C07D501/04;C07D501/06;C07D501/22;C07D501/24;C07D501/26;C07D501/34 主分类号 C07D501/20
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