发明名称 IMIDAZO(1,2-A)QUINOLINE DERIVATIVES
摘要 Novel imidazo[1,2-a]quinolines of the formula <IMAGE> I wherein R is selected from the group consisting of alkyl of 1 to 8 carbon atoms, thienyl, pyridyl and phenyl optionally substituted with at least one member of the group consisting of halogen, alkyl of 1 to 5 carbon atoms and alkoxy of 1 to 5 carbon atoms, R1 and R2 are individually selected from the group consisting of hydrogen, halogen, alkyl and alkoxy of 1 to 8 carbon atoms,s cyclohexyl, -NO2 and phenoxy, R3 is selected from the group consisting of alkoxy and alkylthio of 1 to 8 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts having a remarkable anxiolytic activity and a hypnotic activity and their preparation.
申请公布号 EP0062580(B1) 申请公布日期 1985.11.06
申请号 EP19820400590 申请日期 1982.03.31
申请人 ROUSSEL-UCLAF 发明人 BARNES, ALAN CHARLES;ROBSON, PETER ANDREW
分类号 C07D471/00;A61K31/47;A61P25/20;C07D215/38;C07D471/04 主分类号 C07D471/00
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