摘要 |
<p>Novel 2,3,4,5-tetrahydro-1H-pyridoindole derivatives of the formula R'' W3, wherein R'' is < IMG > k is 1 or 2; X and Y are each independently H, F, Cl, Br, OCH3, CH3 or CH2CH3; W3 is -(CH2)n-NR5R6; n is 1 to 9; R5 taken separately is hydrogen; R6 taken separately is (C1-C8)alkanoyl or (C1-C7) alkoxycarbonyl; and R5 and R6 taken together are < IMG > wherein r is 3 to 5; or a pharmaceutically acid addition salt thereof are prepared by various standard reactions. The compounds are useful as neuroleptic agents in the treatment of mental disorders and illnesses.</p> |