发明名称 PROCESS FOR PREPARING HEXAHYDRO-TRANS-PYRIDOINDOLE
摘要 Title compds. (I; X and Y are independently H, F; R= C1-3 alkanoyl, C2-3 alkoxycarbonyl, (substituted benzoyl or phenyl sulfonyl; m = 2-9), their racemates, enantiomers, and salts, were prepd. from V. I was useful as tranquilizers, having fewer side-effects than the commonly used drugs. Thus, lg trans-I reacted with 0.723 g γ-bromo-butyronitrile and the product was reduced with LiAlH4 to give 0.498 g I.
申请公布号 KR840000914(B1) 申请公布日期 1984.06.28
申请号 KR19800003000 申请日期 1980.07.28
申请人 PFIZER INC. 发明人 WELCH WILLARD MCKOWAN;HARBERT CHARLES ARMON
分类号 A61K31/435;A61P25/18;A61P25/20;C07D471/04;(IPC1-7):C07D471/04 主分类号 A61K31/435
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