发明名称 MELLANPRODUKT FOR FRAMSTELLNING AV IMIDAZO /1,5-A/ /1,4/ DIAZEPINDERIVAT
摘要 Imidazo[1,5-a][1,4]diazepine compounds of the formula <IMAGE> in which the symbols <IMAGE>, A, R1, R2 and R3 have the meaning given in Claim 1, analogues thereof as are defined in Claims 2 to 4, and pharmaceutical utilisable acid addition salts of these compounds have useful muscle-relaxant, sedative and anti-convulsive properties. They are particularly suitable for the preparation of injection solutions on account of the good water solubility of their acid addition salts. The compounds are prepared by dehydrogenation of the corresponding 3a,4-dihydro derivatives and optional N-oxidation, reduction or reaction with ethylene oxide or propylene oxide.
申请公布号 SE433080(B) 申请公布日期 1984.05.07
申请号 SE19790002667 申请日期 1979.03.23
申请人 F HOFFMANN-LA ROCHE & CO AG 发明人 R I * FRYER;A * WALSER
分类号 C07D243/16;A61K31/55;A61K31/551;A61K31/5517;A61P21/02;A61P25/20;C07D233/54;C07D233/64;C07D249/08;C07D487/04;C07D487/14;C07D495/04;C07D495/14;C07D498/14;C07D498/22;C07F9/645;C07F9/6561;F16L59/02;(IPC1-7):07D487/04;07D495/16 主分类号 C07D243/16
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