发明名称 |
ANALOGIFREMGANGSMAADE TIL FREMSTILLING AF 4'-DEOXYDAUNOMYCIN |
摘要 |
<p>The novel compounds, 4'-deoxy-daunomycin and 4'-deoxy-adriamycin, as well as derivatives thereof are useful as anti-tumor antibiotics. These compounds are prepared by condensing the corresponding aglycone with a novel trifluoracetyl protected reactive halo sugar which is 2,3,4,6-tetradeoxy-3-trifluoroacetamido-L-threo-hexopyranosyl chloride.</p> |
申请公布号 |
DK146626(C) |
申请公布日期 |
1984.04.30 |
申请号 |
DK19760004260 |
申请日期 |
1976.09.22 |
申请人 |
FARMITALIA CARLO ERBA S.P.A. |
发明人 |
PENCO SERGIO;ARCAMONE FEDERICO;MARCO AURELIO DI |
分类号 |
A61K31/35;A61K31/351;A61K31/65;A61K31/704;A61P35/00;A61P35/02;C07D309/14;C07H13/04;C07H15/252;(IPC1-7):C07D309/14 |
主分类号 |
A61K31/35 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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