发明名称 SUBSTITUERADE FENYLACETYLENER JEMTE SETT FOR DERAS FRAMSTELLNING
摘要 The compounds of formula I, in which R<1> is H, alkyl, aralkyl or diaralkyl, R<2> is H or a halogen and R<3> is H, alkyl, aralkyl, aryl, aryloxy, benzoyl or 2-thienocarbonyl, R<2> and R<3> not being simultaneously H, are obtained by halogenation of a ketone of formula II, followed by dehydrohalogenation of the intermediate halogenated derivative of formula III by means of a strong base. The compounds of formula I are useful as intermediates for the preparation of pharmaceutically active compounds. <IMAGE>
申请公布号 SE431867(B) 申请公布日期 1984.03.05
申请号 SE19770005840 申请日期 1977.05.17
申请人 CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT 发明人 E * PALOSI;G * HEJA;D * KORBONITS;C * GONCZI;P * KISS;R
分类号 C07C43/285;C07C1/00;C07C1/24;C07C1/30;C07C11/22;C07C15/48;C07C17/00;C07C17/18;C07C17/25;C07C25/02;C07C25/18;C07C25/24;C07C41/00;C07C45/00;C07C45/63;C07C45/65;C07C49/76;C07C67/00;C07D333/22;(IPC1-7):07C15/48 主分类号 C07C43/285
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