发明名称 Sulphonamides.
摘要 <p>Compounds of the formula (I) and salts thereof: &lt;Chemistry id="chema01" num="0001"&gt;&lt;Image id="ia01" he="26" wi="95" file="IMGA0001.TIF" imgContent="chem" imgFormat="TIFF" inline="no" /&gt;&lt;/Chemistry&gt;wnerem: &lt;UnorderedLists id="ula01" listStyle="none"&gt;&lt;ListItem&gt;A is a bond, -CH&lt;Sub&gt;2&lt;/Sub&gt;- or -CH=CH-;&lt;/ListItem&gt;&lt;ListItem&gt;R&lt;Sup&gt;2&lt;/Sup&gt; is hydrogen and R&lt;Sup&gt;1&lt;/Sup&gt; is selected from C&lt;Sub&gt;1-4&lt;/Sub&gt; alkyl, hydroxyl, C&lt;Sub&gt;1-4&lt;/Sub&gt; alkoxy, C&lt;Sub&gt;1-4&lt;/Sub&gt; alkanoyloxy, hydrogen, halogen, nitro, cyano, and amino optionally substituted by one or two C&lt;Sub&gt;1-4&lt;/Sub&gt; alkyl groups or by C&lt;Sub&gt;1-4&lt;/Sub&gt; alkanoyl;&lt;/ListItem&gt;&lt;ListItem&gt;R&lt;Sup&gt;4&lt;/Sup&gt; is C&lt;Sub&gt;1-4&lt;/Sub&gt; alkyl, hydroxy, C&lt;Sub&gt;1-4&lt;/Sub&gt; alkoxy, C&lt;Sub&gt;1-4&lt;/Sub&gt; alkanoyloxy or n&lt;Sup&gt;i&lt;/Sup&gt;trato;&lt;/ListItem&gt;&lt;ListItem&gt;R&lt;Sub&gt;2&lt;/Sub&gt;N is 1-piperidyl, morpholino or 4-methyl-1-piperazyl, optionally substituted by one or two methyl groups in the 2-, 4- or 6- positions as apt, or 1-pyrrolidyl substituted by one or two methyl groups.&lt;/ListItem&gt;&lt;ListItem&gt;m is 0 or 1; and&lt;/ListItem&gt;&lt;ListItem&gt;n is 0 to 3&lt;/ListItem&gt;&lt;/UnorderedLists&gt; a process for their preparation and compositions containing them.</p>
申请公布号 EP0076072(A2) 申请公布日期 1983.04.06
申请号 EP19820304929 申请日期 1982.09.20
申请人 BEECHAM - WUELFING GMBH & CO. KG 发明人 JOZIC, LJERKA
分类号 C07D295/12;A61K31/40;A61P9/06;C07D207/06;C07D211/14;C07D295/13;(IPC1-7):07D295/12;07D211/14;61K31/395;07D207/06 主分类号 C07D295/12
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