发明名称 PYRIMIDONE DERIVATIVE
摘要 The present inventions provides compound of formula (II): <CHEM> and their pharmaceutically acceptable salts which are useful as histamine H1-antagonists. In formula (II) R is C1-4 alkyl, and R<2> is C3-4 alkoxy, halogen, oramino: R<3> is a C1-3 alkylene group; and R<4> is a 3-pyridyl, N-oxo-3-pyridyl, 6-methyl-3-pyridyl, N-oxo-6-methyl-3-pyridyl or 6-hydroxymethyl-3-pyridyl group.
申请公布号 JPS588080(A) 申请公布日期 1983.01.18
申请号 JP19820110568 申请日期 1982.06.26
申请人 SMITH KLINE & FRENCH LAB LTD 发明人 JIYOOJI SHIDONII SATSUCHI
分类号 B41M1/16;A61K31/505;A61K31/506;A61K31/513;A61P11/04;A61P11/08;A61P27/16;A61P37/08;A61P43/00;B41M3/12;C07D213/61;C07D213/65;C07D213/68;C07D213/73;C07D213/76;C07D239/36;C07D401/12;C07D401/14;C07D403/14 主分类号 B41M1/16
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