发明名称 FOERFARANDE FOER FRAMSTAELLNING AV BRONKOSEKRETEROLYTISKA 5,11-DIHYDRO-5H-PYRIDO(2,3-B)(1,5)BENSODIAZEPIN-5-ONER
摘要 Compounds of the formula <IMAGE> wherein R1-is hydrogen, alkyl of 1 to 6 carbon atoms or benzyl; R2-is alkyl of 1 to 6 carbon atoms, cycloalkyl of 5 to 7 carbon atoms or, together with R1 and the adjacent nitrogen atom, pyrrolidino, piperidino, hexamethyleneimino, morpholino or N'-methyl-piperazino, where each of the heterocycles may have one or two alkyl of 1 to 3 carbon atoms or one or two methoxy substituents attached thereto; R3,-R4 and R5 are each hydrogen or methyl; R6-is alkyl of 1 to 4 carbon atoms; and A-is alkylene of 2 to 4 carbon atoms; AND NON-TOXIC, PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF; THE COMPOUNDS AS WELL AS THEIR SALTS ARE USEFUL AS BRONCHOSPASMOLYTICS AND BRONCHOSECRETOLYTICS.
申请公布号 FI62086(C) 申请公布日期 1982.11.10
申请号 FI19770002772 申请日期 1977.09.20
申请人 DR KARL THOMAE G M B H 发明人 SCHMIDT GUENTHER;PUESCHMANN SIGFRID;ENGELHARDT GUENTHER
分类号 A61K31/55;A61K31/551;A61P11/08;A61P11/10;C07D213/80;C07D471/04;(IPC1-7):C07D471/04 主分类号 A61K31/55
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