发明名称 Phenicol antibacterials
摘要 Disclosed herein are phenicol derivatives of formula I where the variables are as defined herein. Also disclosed is their use for the treatment of infections in mammals, pharmaceutical compositions containing the compounds, and methods for the preparation of these compounds. Specific examples of the compounds of formula I are N-((1R,2S)-3-fluoro-1-hydroxy-1-(4-(6-(methyl-sulfonamidomethyl)pyridin-3-yl)phenyl)propan-2-yl)methanesulfonamide and N-((1R,2S)-1-(4-(2-(1-aminoethyl)thiazol-5-yl)phenyl)-3-fluoro-1-hydroxypropan-2-yl)-2,2-difluoroacetamide.
申请公布号 NZ630099(A) 申请公布日期 2016.08.26
申请号 NZ20130630099 申请日期 2013.03.01
申请人 ZOETIS SERVICES LLC 发明人 DUCLOS BRIAN A.;BILLEN DENIS;KYNE GRAHAM M.;SHEEHAN SUSAN M.K.;JOHNSON TIMOTHY A.;VAIRAGOUNDAR RAJENDRAN;HABER-STUK ANDREA K.;EWIN RICHARD A.;CURTIS MICHAEL;JOHNSON PAUL D.;GOODWIN RICHARD M.
分类号 C07D333/20;A61K31/4245;A61K31/427;A61K31/4418;A61K31/4439;A61K31/4995;C07D213/38;C07D239/26;C07D241/12;C07D271/06;C07D277/28;C07D285/12;C07D401/06;C07D413/06;C07D417/06 主分类号 C07D333/20
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