PROCESS FOR THE PREPARATION OF 2-AMINO-BENZYLAMINES

摘要

2-amino-benzylamine The invention relates to a new process for the preparation of 2-amino-benzylamine derivatives having valuable pharmacological properties, in particular a secretolytic and/or antitussive activity. The process comprises the reaction of the corresponding 2-amino-benzyl alcohol with an appropriate amine, either the amino group being acylated or the reaction being performed in the presence of an organic acid. Examples of the proparation of certain 2-amino-benzylamine by means of the new process are given.