发明名称 |
Use of 6-chloro-3-methyl-1H-2,3,4,5-tetrahydro-3-benzazepine-n-oxide, as a prodrug |
摘要 |
6-Chloro-3-methyl-1H-2,3,4,5-tetrahydro-3-benzazepine-N-oxide is prepared by mild oxidation of the corresponding amine. It has been found to have prolonged alpha 2-antagonistic or antihypertensive activity.
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申请公布号 |
US4686218(A) |
申请公布日期 |
1987.08.11 |
申请号 |
US19850696377 |
申请日期 |
1985.01.30 |
申请人 |
SMITHKLINE BECKMAN CORPORATION |
发明人 |
DEMARINIS, ROBERT M.;STRAUB, KENNETH M. |
分类号 |
A61K31/55;A61P9/12;A61P25/02;C07D223/16;(IPC1-7):A61K31/55 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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