发明名称 Use of 6-chloro-3-methyl-1H-2,3,4,5-tetrahydro-3-benzazepine-n-oxide, as a prodrug
摘要 6-Chloro-3-methyl-1H-2,3,4,5-tetrahydro-3-benzazepine-N-oxide is prepared by mild oxidation of the corresponding amine. It has been found to have prolonged alpha 2-antagonistic or antihypertensive activity.
申请公布号 US4686218(A) 申请公布日期 1987.08.11
申请号 US19850696377 申请日期 1985.01.30
申请人 SMITHKLINE BECKMAN CORPORATION 发明人 DEMARINIS, ROBERT M.;STRAUB, KENNETH M.
分类号 A61K31/55;A61P9/12;A61P25/02;C07D223/16;(IPC1-7):A61K31/55 主分类号 A61K31/55
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