发明名称 PROCEDIMIENTO PARA PREPARAR DERIVADOS DE ANILIDAS.
摘要 <p>1500576 Amides CIBA-GEIGY AG 8 April 1975 [9 April 1974 7 March 1975] 14379/75 Heading C2C The invention comprises compounds of the formula wherein R 1 represents a halogen atom or an alkyl or alkoxy group of 1 to 4 carbon atoms, R 2 represents a hydrogen or halogen atom, an alkyl group of 1 to 3 carbon atoms or an alkoxy group of 1 to 4 carbon atoms, R 3 represents a hydrogen atom, or a methyl or ethyl group, R 4 represents an alkyl group of 1 to 6 carbon atoms unsubstituted or substituted by cyano (-CN) or rhodano (-SCN), an alkenyl group of 2 to 5 carbon atoms or a cycloalkyl group of 3 to 7 carbon atoms, R 5 represents a hydrogen or halogen atom, or an alkyl group of 1 to 3 carbon atoms, and R 6 represents a hydrogen atom or a methyl group, the total number of carbon atoms in the substituents R 1 , R 2 , R 5 and R 6 not exceeding 8. The compounds may be prepared by acylating a compound of the formula with a compound of the formula HO-CO-R 4 or with a reactive derivative thereof, or by converting a compound of the formula with butyl lithium or sodium hydride into the corresponding alkali salt which is then reacted with a compound of the formula where Hal is halogen or another easily removable radical, or by reacting the compound of Formula IV with Hal-CH(CH 3 )-COOR 3 in the presence of an alkali carbonate.</p>
申请公布号 ES436384(A1) 申请公布日期 1977.04.01
申请号 ES19840004363 申请日期 1975.04.08
申请人 CIBA-GEIGY, A.G. 发明人
分类号 A01N47/20;A01N37/22;A01N37/34;A01N37/46;A01N47/48;A01N53/12;A61K31/24;C07C67/00;C07C231/00;C07C231/02;C07C231/10;C07C233/38;C07C233/88;C07C237/06;C07C253/00;C07C255/27;C07C325/00;C07C331/14;(IPC1-7):01N/ 主分类号 A01N47/20
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