发明名称 Enzyme inhibitors
摘要 The invention relates to an intermediate of formula (VI) <CHEM> or a protected derivative thereof, wherein Q is hydrogen or a carboxyl protecting group and Q' is a protecting group. Such intermediates are useful for the preparation of amidino sulphone derivatives which, in turn, have use as selective inhibitors of inducible nitric oxide synthase.
申请公布号 AU692892(B2) 申请公布日期 1998.06.18
申请号 AU19950028917 申请日期 1995.06.14
申请人 THE WELLCOME FOUNDATION LIMITED 发明人 HAROLD FRANCIS HODSON;RICHARD MICHAEL JOHN PALMER;DAVID ALAN SAWYER;RICHARD GRAHAM KNOWLES;KARL WITOLD FRANZMANN;MARTIN JAMES DRYSDALE;STEVEN SMITH;PATRICIA IFEYINWA DAVIES;HELEN ALICE REBECCA CLARK;BARRY GEORGE SHEARER
分类号 A61K31/00;A61K;A61K31/195;A61K31/198;A61P5/00;A61P9/00;A61P43/00;C07C;C07C257/14;C07C315/02;C07C317/02;C07C317/48;C07C317/50;C07C323/60;C07C327/58;(IPC1-7):C07C317/48 主分类号 A61K31/00
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