Quinolinone derivatives as PARP and TANK inhibitors
摘要
The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, R7, n, m and X have defined meanings.
申请公布号
AU2008223793(A1)
申请公布日期
2008.09.12
申请号
AU20080223793
申请日期
2008.03.07
申请人
JANSSEN PHARMACEUTICA NV
发明人
ELISABETH THERESE JEANNE PASQUIER;JAMES EDWARD STEWART DUFFY;XAVIER MARC BOURDREZ;ANDREW PATE OWENS;EDDY JEAN EDGARD FREYNE;VIRGINIE SOPHIE PONCELET;BRUNO ROUX;JACQUELINE ANNE MACRITCHIE;PATRICK RENE ANGIBAUD;LAURENCE FRANCOISE BERNADETTE MARCONNET-DECRANE;PIERRE-HENRI STORCK;CHRISTOPHE MEYER;LAURENCE ANNE MEVELLEC;JORGE EDUARDO VIALARD;CHRISTOPHE DENIS ADELINET;ISABELLE NOELLE CONSTANCE PILATTE