发明名称 PIPERIDYINDOLES AS SEROTONIN RECEPTOR LIGANDS
摘要 A pharmaceutical compound of the formula (I) in which R<1> and R<2> are each hydrogen or C1-6 alkyl, R<3> is -SR<10>, -SOR<10>, -SO2R<10>, -COR<10>, -CH2OH or -CONHR<11>, where R<10> is C1-6 alkyl and R<11> is hydrogen or C1-6 alkyl, R<4>, R<5>, R<6> and R<7> are each hydrogen or C1-6 alkyl, provided that at least one of R<4>, R<5>, R<6> and R<7> is C1-6 alkyl, R<8> and R<9> are each hydrogen, halo, C1-6 alkyl or cyano, n is 0 or 1 and m is 2 or 3, x is a (a) or (b), and y is (c) or (d), wherein R<12> and R<13> are each hydrogen, C1- alkyl, cyclopropyl or cyclopropyl-C1-6 alkyl; and salts thereof.
申请公布号 WO0187881(A1) 申请公布日期 2001.11.22
申请号 WO2001US11744 申请日期 2001.05.04
申请人 ELI LILLY AND COMPANY;FAIRHURST, JOHN;GALLAGHER, PETER 发明人 FAIRHURST, JOHN;GALLAGHER, PETER
分类号 A61K31/4709;A61K31/5415;A61P1/00;A61P1/08;A61P3/04;A61P9/10;A61P9/12;A61P15/10;A61P25/00;A61P25/04;A61P25/08;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/32;A61P25/34;A61P25/36;A61P43/00;C07D401/14;C07D417/14;(IPC1-7):C07D417/14;A61K31/54;A61K31/475;A61K31/445 主分类号 A61K31/4709
代理机构 代理人
主权项
地址