发明名称 BENZODIAZEPHINE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY
摘要 T1105Y BENZODIAZEPINE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY Compounds of formula (I), and salts and prodrugs thereof (I) wherein: R1 represents optionally substituted C1-6alkyl or C3-7cycloalkyl; R2 represents an optionally substituted phenyl or pyridyl group; R3 represents C1-6 alkyl or halo; R4 represents C3-7 cycloalkyl; x is 0, 1, 2 or 3; are CCK and/or gastrin antagonists. They and compositions thereof are therefore useful in therapy.
申请公布号 CA2068355(A1) 申请公布日期 1992.11.15
申请号 CA19922068355 申请日期 1992.05.11
申请人 MERCK SHARP & DOHME LIMITED 发明人 CHAMBERS, MARK S.;FLETCHER, STEPHEN R.;MATASSA, VICTOR G.
分类号 A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P25/00;A61P25/02;C07D243/14;C07D243/24;C07D401/12;C07D403/12;C07D417/12;C07D521/00;(IPC1-7):C07D243/14;C07D405/12;C07D409/12;C07F9/645;A61K31/675 主分类号 A61K31/55
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