发明名称 |
BENZODIAZEPHINE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY |
摘要 |
T1105Y BENZODIAZEPINE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY Compounds of formula (I), and salts and prodrugs thereof (I) wherein: R1 represents optionally substituted C1-6alkyl or C3-7cycloalkyl; R2 represents an optionally substituted phenyl or pyridyl group; R3 represents C1-6 alkyl or halo; R4 represents C3-7 cycloalkyl; x is 0, 1, 2 or 3; are CCK and/or gastrin antagonists. They and compositions thereof are therefore useful in therapy.
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申请公布号 |
CA2068355(A1) |
申请公布日期 |
1992.11.15 |
申请号 |
CA19922068355 |
申请日期 |
1992.05.11 |
申请人 |
MERCK SHARP & DOHME LIMITED |
发明人 |
CHAMBERS, MARK S.;FLETCHER, STEPHEN R.;MATASSA, VICTOR G. |
分类号 |
A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P25/00;A61P25/02;C07D243/14;C07D243/24;C07D401/12;C07D403/12;C07D417/12;C07D521/00;(IPC1-7):C07D243/14;C07D405/12;C07D409/12;C07F9/645;A61K31/675 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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