发明名称 Gaba-agonistic imidazo(4,5-c)pyridines useful as pharmaceuticals
摘要 Imidazo(4,5-c)pyridines of the formula <IMAGE> wherein X is O, S or NH; Y is -NR2-CH=N- or -N=CH-NR2-; R1 is 1-benzothienylmethyl, naphthylmethyl, or benzyl which is mono- or di-substituted by F, Cl, NO2, CF3 or a combination thereof, and; R2 is alkyl of 1-4 C atoms or cyclopropylmethyl, or a physiologically acceptable acid addition salt thereof, have valuable pharmacological activity, e.g., as GABA agonists.
申请公布号 US4654350(A) 申请公布日期 1987.03.31
申请号 US19860873560 申请日期 1986.06.12
申请人 MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG 发明人 IRMSCHER, KLAUS;SAIKO, OTTO;MINCK, KLAUS-OTTO;WOLF, HANS-PETER
分类号 A61K31/435;A61P3/04;A61P25/08;A61P39/02;C07D471/04;(IPC1-7):A61K31/44 主分类号 A61K31/435
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