发明名称 PHENYLPIPERAZINE DERIVATIVES OF HETARYLPHENOLS AND HETARYLANILINES, THEIR PREPARATION, AND THERAPEUTIC AGENTS CONTAINING THESE COMPOUNDS
摘要 <p>Novel phenylpiperazinylpropane and -butane derivatives of hetarylphenols and hetarylanilines of the formula < IMG > where R1 is hydrogen or alkyl of 1 to 4 carbon atoms, R2 is hydrogen, halogen, alkyl of 1 to 4 carbon atoms or alkoxy where alkyl is of 1 to 3 carbon atoms, the phenyl ring can be monosubstituted or disubstituted by R2, X is oxygen or an NH group, and the heterocyclic structure Het. is 1,3,4oxadiazolyl, triazolyl, imidazolyl or pyrazolyl, and their physiologically tolerated addition salts with acids, processes for their preparation, and pharmaceutical formulations which contain these compounds and exhibit predominantly sedative, neuroleptic and hypotensive properties.</p>
申请公布号 CA1187878(A) 申请公布日期 1985.05.28
申请号 CA19820394179 申请日期 1982.01.14
申请人 BASF AKTIENGESELLSCHAFT 发明人 THIEME, PETER C.;STEINER, GERD;ROHR, WOLFGANG;LENKE, DIETER;GRIES, JOSEF;WEIFENBACH, HARALD;TESCHENDORF, HANS-JUERGEN;HOFMANN, HANS P.;KREISKOTT, HORST
分类号 C07D249/08;A61K31/495;A61K31/496;A61P9/02;A61P11/00;A61P25/20;C07D231/12;C07D233/60;C07D233/61;C07D271/10;C07D295/06;C07D295/067;C07D295/096;C07D521/00;(IPC1-7):C07D295/04;C07D403/12 主分类号 C07D249/08
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