发明名称 ANTIBACTERIAL QUINAZOLINE-4(3H)-ONE DERIVATIVES
摘要 The invention relates to antibacterial compounds of formula I, wherein R1 is H or halogen; R2 is the group M; R3 is H or halogen; M is MA or MB wherein A is a bond or C≡C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, hydroxyalkyl, 1,2-dihydroxyethyl, dialkylamino, 1-hydroxymethyl-cycloprop-1-yl, 1-((dimethylglycyl)oxy)methyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, morpholin-4-ylalkyl or morpholin-4-ylalkoxy; and R1B is a group as defined in claim 1; and salts thereof.
申请公布号 EP3143007(A1) 申请公布日期 2017.03.22
申请号 EP20150722212 申请日期 2015.05.13
申请人 Actelion Pharmaceuticals Ltd 发明人 GAUVIN, Jean-Christophe;SURIVET, Jean-Philippe;CHAPOUX, Gaëlle;MIRRE, Azely
分类号 C07D239/90;A61K31/517;A61P31/04 主分类号 C07D239/90
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