发明名称 2,5-DISUBSTITUTED CYCLOPENTANECARBOXYLIC ACIDS AND THEIR USE
摘要 The present application relates to novel 2,5-disubstituted cyclopentanecarboxylic acid derivatives, to processes for preparation thereof, to the use thereof alone or in combinations for treatment and/or prevention of diseases and to the use thereof for production of medicaments for treatment and/or prevention of diseases, especially for treatment and/or prevention of respiratory, pulmonary and cardiovascular disorders.
申请公布号 US2017022171(A1) 申请公布日期 2017.01.26
申请号 US201515301392 申请日期 2015.03.31
申请人 Bayer Pharma Aktiengesellschaft 发明人 BECK Hartmut;LI Volkhart Min-Jian;CANCHO GRANDE Yolanda;TIMMERMANN Andreas;BROHM Dirk;JÖRISSEN Hannah;BOGNER Pamela;GERISCH Michael;LANG Dieter
分类号 C07D253/08;A61K31/53;C07D413/12;A61K45/06 主分类号 C07D253/08
代理机构 代理人
主权项 1. A compound of the formula (I) in which A is —O— or —S—, R1 is straight-chain or branched (C3-C7)-alkyl or a group of the formula in which* indicates the linkage to A,n is the number 1, 2 or 3,Cy is (C3-C6)-cycloalkyl, R3A is hydrogen, fluorine, chlorine, cyano, methyl, difluoromethyl, trifluoromethyl, methoxy, trifluoromethoxy, (trifluoromethyl)sulphanyl, methoxycarbonylamino or 2-oxo-1,3-oxazolidin-3-yl, andR3B is hydrogen, fluorine, chlorine, methyl or trifluoromethyl, and R2 is hydrogen, fluoromethyl, methyl, difluoromethyl or trifluoromethyl, or a salt, solvate or solvate of a salt of this compound.
地址 Berlin DE