NOVEL SUBSTITUTED BICYCLIC COMPOUNDS AS BROMODOMAIN INHIBITORS
摘要
The invention relates to substituted bicyclic compounds, which are useful for inhibition of BET protein function by binding to bromodomains, pharmaceutical compositions comprising these compounds, and use of the compounds and compositions in therapy.
申请公布号
EP3010917(A4)
申请公布日期
2017.01.25
申请号
EP20140822480
申请日期
2014.06.20
申请人
Zenith Epigenetics Corp.
发明人
LIU, Shuang;QUINN, John, Frederick;DUFFY, Bryan, Cordell;WANG, Ruifang;JIANG, May, Xiaowu;MARTIN, Gregory, Scott;ZHAO, He;ELLIS, Michael;WAGNER, Gregory, Steven;YOUNG, Peter, Ronald