| 发明名称 |
CYCLIC VINYLOGOUS AMIDES AS BROMODOMAIN INHIBITORS |
| 摘要 |
Cyclic vinylogous amides of Formula I are disclosed The compounds are useful for treating diseases that arise from inappropriate activity of proteins containing an acetyl-lysine. The compositions comprise a genus of cyclic vinylogous amides that are inhibitors of bromodomain. |
| 申请公布号 |
EP3038612(A4) |
申请公布日期 |
2017.01.11 |
| 申请号 |
EP20140839424 |
申请日期 |
2014.08.29 |
| 申请人 |
Icahn School of Medicine at Mount Sinai |
发明人 |
ZHOU, Ming-Ming;OHLMEYER, Michael;VINCEK, Adam;ZAWARE, Nilesh |
| 分类号 |
C07D213/75;A61K31/122;A61P35/00;A61P37/00;C07D209/40;C07D213/76;C07D215/38;C07D249/06 |
主分类号 |
C07D213/75 |
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