发明名称 TETRACYCLIC COMPOUNDS
摘要 FIELD: organic chemistry.SUBSTANCE: invention relates to organic chemistry, specifically to a particular 9-ethyl-6,6-dimethyl-8-(4-morpholine-4-yl-piperidine-1-yl)-11-oxo-6,11-dihydro-5H-dihydro-5H-benzo [b]carbazole-3-carbonitrile . Invention also relates to a medicament, an ALK inhibitor and pharmaceutical composition based on particular benzo-carbazole derivative.EFFECT: novel benzo-carbazole derivatives which are useful in treating cancer are obtained.7 cl, 49 tbl, 1218 ex
申请公布号 RU2585622(C2) 申请公布日期 2016.05.27
申请号 RU20110154150 申请日期 2010.06.09
申请人 CHUGAI SEJYAKU KABUSIKI KAJSYA 发明人 KINOSITA KAZUTOMO;ASOKH KOKHSUKE;FURUITI NORIYUKI;ITO TOSIYA;KAVADA KHATSUO;ISII NOBUYA;SAKAMOTO KHIROSI;KHONG VOOSANG;PARK MINDZEONG;ONO ESIYUKI;KATO YASUKHARU;MORIKAMI KENDZI;EMURA TAKASI;OIKAVA NOBUKHIRO
分类号 C07D209/88;A61K31/343;A61K31/403;A61P35/00;C07D307/92;C07D333/76;C07D401/06;C07D405/12;C07D471/04;C07D491/107 主分类号 C07D209/88
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