发明名称 PROCESS FOR PREPARING PRASUGREL, INTERMEDIATE COMPOUND IN A CRYSTALLINE FORM AND PROCESS FOR PREPARING THE SAME
摘要 The object of the present invention is a process for preparing the 2-acetoxy-5-(2-fluor-α-cyclopropyl-carbonyl-benzyl)-4,5,6,7-tetrahydro-4H-tieno[3,2-c]pyridine (prasugrel) of the formula (I)starting from 5-trityl-4,5,6,7-tetrahydro-tieno[3,2-c]pyridine of the formula (VI)in a crystalline form I. Further objects of the present invention are said novel crystalline form I of the formula (VI) and a process for preparing the same.
申请公布号 EA023057(B1) 申请公布日期 2016.04.29
申请号 EA20120090535 申请日期 2010.12.21
申请人 EGIS GYOGYSZERGYAR NYILANOSAN MUKOEDO RESZVENYTARSASAG 发明人 PORCS-MAKKAY MARTA;VOLK BALAZS;GREGOR TAMAS;BARKOCZY JOZSEF;MEZEI TIBOR;BRODA JUDIT;NYULASI BALINT;RUZSICS GYOERGY;MOLNAR ENIKO;DEBRECZENI JOZSEF;NAGY KALMAN;PANDUR ANGELA;SZENT-KIRALLYI ZSUZSANNA
分类号 C07D495/04 主分类号 C07D495/04
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