发明名称 Insecticidal triazines and pyrimidines
摘要 The present invention describes novel triazines, their related pyrimidines and their use in controlling insects. This invention also includes new synthetic procedures, intermediates for preparing the compounds, pesticide compositions containing the compounds, and methods of controlling insects using the compounds.
申请公布号 US9321735(B2) 申请公布日期 2016.04.26
申请号 US201113810703 申请日期 2011.07.20
申请人 Vestaron Corporation 发明人 Kennedy Robert M.;Steinbaugh Bruce A.
分类号 A61K31/53;A61K31/505;A61K31/506;A01N43/54;A01N43/66;C07D239/49;A01N43/68;A01N43/84;C07D239/48;C07D251/48;C07D401/12;C07D403/12;C07D409/12;C07D413/12;C07D405/12 主分类号 A61K31/53
代理机构 Honigman Miller Schwartz & Cohn LLP 代理人 Honigman Miller Schwartz & Cohn LLP ;Wootton Thomas A.;O'Brien Jonathan P.
主权项 1. A method of using the compounds of Formula (I), wherein: Y is N or CR1; R1, is —H, Halo or —C1-C4 alkyl; Z is -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C6 alkylC6cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, X, is —H, —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, —NRiRj or —C1-C8 alkylNRiRj; R2 and R3 are independently —H or —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, and —C1-C8 alkylNRiNj, but R2 and R3 are not both H; Ri and Rj are independently —H, or —C1-C8 alkyl; wherein heterocyclic is a 5-10 member cyclic or bicyclic aromatic or saturated —C1-C8 cycloaliphatic ring moiety containing 1, 2, or 3 heteroatoms selected from N, O, or S; wherein aryl, —C3-C8 cycloalkyl and heterocyclic are optionally independently substituted with one to five substituents independently selected from -halo, —CN, —OH, —OCH2CH═CHCl, —C1-C6 alkyl, —O—C1-C6 alkyl, or —S—C1-C6 alkyl; and at each occurrence alkyl, is optionally substituted with 1-5 halo, —CN, or —OH to control and inhibit: insects, mites and nematodes, comprising applying an insect-inhibiting amount of a compound of Formula I to the locus, area to be protected or directly on the insects, mites and nematodes.
地址 Kalamazoo MI US
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