发明名称 (r)-3-(e)-2-(pirrolidin-33-il)vinil)-5-(tetra-hidropiran-4-ilóxi)piridina, seus sais, suas sínteses e seus usos como ligantes para receptores acetilcolinérgico nicotínicos
摘要 The present invention relates to the hemi-galactarate, oxalate and di-p-toluoyl-D-tartrate salt forms of (R)-3-((E)-2-(pyrrolidin-3-yl)vinyl)-5-(tetrahydropyran-4-yloxy)pyridine or hydrates or solvates thereof, compositions comprising these salt and their use for treating or preventing a NNR mediated disorder.
申请公布号 BRPI0922630(A2) 申请公布日期 2016.01.05
申请号 BR2009PI22630 申请日期 2009.11.30
申请人 TARGACEPT, INC 发明人 DANIEL YOHANNES;GARY MAURICE DULL;GREGORY J. GATTO;JOHN GENUS;JOSEPH PIKE MITCHENER, JR.;JULIO A. MUNOZ;NIKOLAI FEDOROV;PHILIP S. HAMMOND;PIETER ALBERT OTTEN;SCOTT R. BREINING;SRINIVISA RAO AKIREDDY;TIMOTHY J. CUTHBERTSON
分类号 C07D405/14;A61K31/4439;A61P25/00 主分类号 C07D405/14
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