发明名称 VERFAHREN ZUR HERSTELLUNG VON LAMOTRIGIN UND DESSEN ZWISCHENPRODUKT 2,3-DICHLORBENZOYLCHLORID
摘要 <p>A method for preparing 3,5-diamino-6-(2,3-dichlorophenyl)-1,2,4-triazine, commonly known as lamotrigine, is disclosed. A method of preparing the intermediate, 2,3-dichlorobenzoyl chloride, by photochlorination of 2,3-dichlorobenzotrichloride followed by hydrolysis is also disclosed. The intermediate may then be used in the preparation of lamotrigine.</p>
申请公布号 DE602007003830(D1) 申请公布日期 2010.01.28
申请号 DE20076003830T 申请日期 2007.05.30
申请人 CALAIRE CHIMIE SAS 发明人 VAN DEYNSE, DIRK;BELMANS, MARC;BOERS, FRANK;DUMUR, MICHEL;LACONI, ALAIN
分类号 C07D253/06 主分类号 C07D253/06
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