发明名称 A PROCESS FOR THE PREPARATION OF DIPHENOXYLATE HYDROCHLORIDE
摘要 <p>The present invention relates to an improved process for the preparation of diphenoxylate hydrochloride of the formula (I) by condensing 4-Bromo-2,2-diphenylbutanenitrile ( II) and Ethyl 4-phenylpiperidine-4-carboxylate (III) in aqueous medium under basic conditions in the presence of a catalyst. This invention also relates to an improved method for purification of the diphenoxylate hydrochloride.</p>
申请公布号 IN5359CH2012(A) 申请公布日期 2015.08.14
申请号 IN2012CH05359 申请日期 2012.12.22
申请人 HYGRO CHEMICALS PHARMTEK PVT. LTD 发明人 DR. D S IYENGAR;DR. ANIL SAIKIA;T M NIRANJAN
分类号 C07D211/00 主分类号 C07D211/00
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