发明名称 Benzoxazole and benzothiazole derivatives, their preparation and their use as synthetic intermediates
摘要 Compounds corresponding to the general formula <IMAGE> in which X represents a nitrogen atom, an oxygen atom or a sulphur atom, Y represents a nitrogen atom, an oxygen atom or a sulphur atom; when X = O or S, then Y = N, and when Y = O or S, then X = N, W represents either a methyl group or a group CH2R' in which R' represents a chlorine atom, a bromine atom or an OR'' group, R'' being a leaving group such as a tosyl group or a mesyl group, Z represents either an iodine atom or a bromine atom or a cyano group or a 1H-tetrazol-5-yl group or a 1-(triphenylmethyl)-1H-tetrazol-5-yl group or a (1,1-dimethylethyl)-1H-tetrazol-5-yl group. Use as intermediates in the synthesis of compounds possessing therapeutic activity.
申请公布号 FR2684377(A1) 申请公布日期 1993.06.04
申请号 FR19910014883 申请日期 1991.12.02
申请人 SYNTHELABO 发明人 CREMER GERARD;MULLER JEAN-CLAUDE
分类号 C07D263/56;C07D263/57;C07D277/66;C07D413/10;C07D417/10 主分类号 C07D263/56
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