发明名称 PROCESS FOR PREPARING APREPITANT
摘要 The present application relates to a process for the preparation of (R)-4-benzyl-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)morpholin-3-one of formula (I), which may be used as an intermediate of aprepitant of formula (V). The present application also relates to a process for the preparation of aprepitant (V).
申请公布号 IN5359CH2013(A) 申请公布日期 2015.09.04
申请号 IN2013CHE5359 申请日期 2013.11.20
申请人 DR. REDDY’S LABORATORIES LIMITED 发明人 JAVED IQBAL;SRINIVAS ORUGANTI;RAJESH KUMAR RAPOLU;VILAS HARESHWAR DAHANUKAR;ELATI RAVI RAM CHANDRASHEKAR;DATTATRAY SHAMRAO METIL;JYOTHIRMAYI NARAM;PALAVI PRAPULLA KUMAR
分类号 C07D413/00 主分类号 C07D413/00
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