发明名称 |
PROCESS FOR PREPARING APREPITANT |
摘要 |
The present application relates to a process for the preparation of (R)-4-benzyl-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)morpholin-3-one of formula (I), which may be used as an intermediate of aprepitant of formula (V). The present application also relates to a process for the preparation of aprepitant (V). |
申请公布号 |
IN5359CH2013(A) |
申请公布日期 |
2015.09.04 |
申请号 |
IN2013CHE5359 |
申请日期 |
2013.11.20 |
申请人 |
DR. REDDY’S LABORATORIES LIMITED |
发明人 |
JAVED IQBAL;SRINIVAS ORUGANTI;RAJESH KUMAR RAPOLU;VILAS HARESHWAR DAHANUKAR;ELATI RAVI RAM CHANDRASHEKAR;DATTATRAY SHAMRAO METIL;JYOTHIRMAYI NARAM;PALAVI PRAPULLA KUMAR |
分类号 |
C07D413/00 |
主分类号 |
C07D413/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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