发明名称 (6S,9aS)-N-BENZYL-6-[(4-HYDROXYPHENYL)METHYL]-4,7-DIOXO-8-({6-[3-(PIPERAZINE-1-YL)AZETIDINE-1-YL]PYRIDINE-2-YL}METHYL)-2-(PROP-2-EN-1-YL)-OCTAHYDRO-1H-PYRAZINO[2,1-c][1,2,4]TRIAZINE-1-CARBOXAMIDE COMPOUND
摘要 Provided is a compound represented by general formula (1) or a pharmaceutically acceptable salt thereof. [In the formula, R1 refers to a C1-6 alkyl group; R2 and R3 are the same or different, and refer to a hydrogen atom or a C1-6 alkyl group; X2, X3, and X4 are the same or different, and refer to a hydrogen atom or halogen atom; and X5 refers to a hydrogen atom, -P(=O)(OH)2.]
申请公布号 WO2015098853(A1) 申请公布日期 2015.07.02
申请号 WO2014JP83932 申请日期 2014.12.22
申请人 EISAI R&D MANAGEMENT CO., LTD.;PRISM PHARMA CO., LTD. 发明人 INOUE SATOSHI;YAMAMOTO YUJI;ISO KENTARO
分类号 C07D487/04;A61K31/53;A61K31/661;A61P11/00;A61P35/00;A61P43/00;C07F9/09 主分类号 C07D487/04
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