2-oxo-piperidinyl derivatives

摘要

The present invention relates to 2-oxo-piperidinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.;

主权项

1. A 2-Oxo-piperidinyl compound of the form according to formula I, or a geometrical isomer, enantiomer, diastereomer or mixture, or a pharmaceutically acceptable salt thereof, wherein
X is either CH or N; Y is either —NR4— or —CH═CH—; with the proviso that X is N when Y is —NR4—;n is an integer selected from 1, 2 or 3; m is 1 or 2;R1 is a substituted or unsubstituted C1-6 alkyl, a substituted or unsubstituted aryl, a substituted or unsubstituted heterocycle, a substituted or unsubstituted C3-8 cycloalkyl; or R1 is a —O—R2 moiety;R2 is a substituted or unsubstituted C1-6 alkyl, a substituted or unsubstituted aryl or a substituted or unsubstituted heteroaryl;R3 is hydrogen, substituted or unsubstituted C1-4 alkyl or halogen; andR4 is hydrogen or C1-4 alkyl.