发明名称 |
TRICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS |
摘要 |
<p>The present invention relates to tricyclic heterocycles which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer.</p> |
申请公布号 |
WO2015095492(A1) |
申请公布日期 |
2015.06.25 |
申请号 |
WO2014US71102 |
申请日期 |
2014.12.18 |
申请人 |
INCYTE CORPORATION;WANG, HAISHENG;SHAO, LIXIN |
发明人 |
WANG, HAISHENG;SHAO, LIXIN;RODGERS, JAMES D.;SHEPARD, STACEY |
分类号 |
C07D471/14;A61K31/43;A61P35/00 |
主分类号 |
C07D471/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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