发明名称 NOVEL POLYMORPHIC FORMS OF 6-(1-METHYL-1H-PYRAZOL-4-YL)-2-{3-[5-(2-MORPHOLIN-4-YL-ETHOXY)-PYRIMIDIN-2-YL]-BENZYL}-2H-PYRIDAZIN-3-ONE DIHYDROGENPHOSPHATE AND PROCESSES OF MANUFACTURING THE SAME
摘要 PROBLEM TO BE SOLVED: To provide novel salt forms of 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2H-pyridazin-3-one, and novel polymorphic forms thereof.SOLUTION: The present invention relates to 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2H-pyridazin-3-one dihydrogenphosphate, its solvates and crystalline modifications thereof.
申请公布号 JP2015028093(A) 申请公布日期 2015.02.12
申请号 JP20140231392 申请日期 2014.11.14
申请人 MERCK PATENT GMBH 发明人 AXEL BECKER;CLEMENS KUEHN;CHRISTOPH SAAL;OLIVER SCHADT;DIETER DORSCH;EVA KRIEGBAUM;FRANK STIEBER;CRISTINA DONINI
分类号 C07D403/14;A61K31/5377;A61K45/00;A61P35/00;A61P35/02;A61P43/00 主分类号 C07D403/14
代理机构 代理人
主权项
地址