发明名称 |
NOVEL POLYMORPHIC FORMS OF 6-(1-METHYL-1H-PYRAZOL-4-YL)-2-{3-[5-(2-MORPHOLIN-4-YL-ETHOXY)-PYRIMIDIN-2-YL]-BENZYL}-2H-PYRIDAZIN-3-ONE DIHYDROGENPHOSPHATE AND PROCESSES OF MANUFACTURING THE SAME |
摘要 |
PROBLEM TO BE SOLVED: To provide novel salt forms of 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2H-pyridazin-3-one, and novel polymorphic forms thereof.SOLUTION: The present invention relates to 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2H-pyridazin-3-one dihydrogenphosphate, its solvates and crystalline modifications thereof. |
申请公布号 |
JP2015028093(A) |
申请公布日期 |
2015.02.12 |
申请号 |
JP20140231392 |
申请日期 |
2014.11.14 |
申请人 |
MERCK PATENT GMBH |
发明人 |
AXEL BECKER;CLEMENS KUEHN;CHRISTOPH SAAL;OLIVER SCHADT;DIETER DORSCH;EVA KRIEGBAUM;FRANK STIEBER;CRISTINA DONINI |
分类号 |
C07D403/14;A61K31/5377;A61K45/00;A61P35/00;A61P35/02;A61P43/00 |
主分类号 |
C07D403/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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